Polebetso hydrokeride pho phohelo
Sinomenine hydrocloride ke motsoako oa lik'hemik'hale o tsoa ho semela sa komporo sa siomenium acutum, e fumanehang ho bochabela. Ke alkaloid eo ka tloaelo e sebelisoang moriana oa China bakeng sa thepa ea eona ea ho ikatisa le e ananeric. Foromo ea hydrochlobile ke letsoai le eketsang tharollo ea komporo le botsitso, e etsa hore e be e loketseng phallo ea merima.
SinOmenine Hydrochloride e ithutile litlamorao tsa eona tsa kalafo maemong a phetetsang joalo ka ramatiki ea Rheumiatoid, ka lebaka la ho putlama ho lefu la mmele le ho fokotsa ho ruruha. E ea sebetsa ka ho thibela tlhahiso ea li-cookline tsa ho ruruha ha li-cractory tsa pottomary le bahlahisi ba bang ba amehang karabelo ea bosholu.
Ntle le litlamorao tsa eona tsa khale-kholo le tsa analges, Sinomenine hydrochloride le tsona li bontšitse bokhoni ba ho ba le Neuroprotection
Lebitso la Ed: (9A, 13a, Ma7,8-Didehydro-4-hydroxy-17-methyl-1-onefinan-1-one, monoh
Nomoro ea CAS: 6080-33-7
Synonyms: Cucoline NSc 76021
Foromo ea limolecular: C19H23no4 • HCL
Foromo ea Mmaro: 365.9
Pustory: ≥98% Crystalline e tiile
Fuubility (ithute ka phapang ea sello)
DMF: 30 mg / ml
DMSO: 30 mg / ml
Ethanol: 5 mg / ml
Pbs (ph 7.2): 5 mg / ml
Tšimoloho: Plamela / Sinotimium actum
Tlhahisoleseling ea ho romella le ea polokelo:
Boloka -20 ° C
Ho tsamaisa: Mocheso oa kamore
Ho tsilatsila: ≥ lilemo tse 4
| Ntho | TLHOKOMELISO | Sephetho |
| Assay (HPLC) | 98.0% | 98.12% |
| Ponahalo | Powder e tšoeu | Ho latela |
| Boholo ba karolo | 98% ho fihlela 80mesh | Ho latela |
| Monko | Tšobotsi | Ho latela |
| Tatso | Tšobotsi | Ho latela |
| Litšobotsi tsa 'mele | ||
| Tahlehelo ea ho omella | ≤0.5% | 0.38% |
| Ash | ≤0.5% | 0.46% |
| Mekhoa e boima | ||
| Litols tse boima (joalo ka pb) | Litekanyetso tsa USP (<10ppm) | <10ppm |
| Arsenic (joalo ka) | ≤2ppm | 0.78ppm |
| Etella pele (PB) | ≤2ppm | 1.13PPM |
| Cadmium (CD) | ≤ppppm | 0.36ppm |
| Mercary (HG) | ≤0.1ppPm | 0.01ppPm |
| Masala a likoluoa | Ha e fumanoe | Ha e fumanoe |
| Kakaretso ea Platecount | Nmt 10000crou / g | 680 CFU / g |
| Tomoso ea tomoso le hlobo | Nmt 100cfu / g | 87 CFU / G |
| E.coli | Nmt 30cfu / g | 10 cfu / g |
| Salmonella | Mpe | Mpe |
| Sephetho | E lumellana le maemo a khoebo | |
Litholoana tse ka sehloohong tsa Sinomen hydrokeride li kenyelletsa:
(1) anti-invi-invi
(2) analgesic: e fana ka phomolo ea bohloko.
(3) Ho itšireletsa: hatella tšebetso ea ts'ireletso ea 'mele.
(4) Anti-Rheamatic: Ho Ts'oarella Rheumatoid Ramatiki.
(5) neuroprotective: e sireletsa lisele tsa methapo.
(6) Anti-Fibrotic: E thibela kapa e fokotsa fibrosis ea lithane.
Sinomenine hydrochloride e sebelisoa haholo libakeng tse latelang:
(1) rheagatogy: kalafo ea Rheumatoid ramatiki.
(2) Tsamaiso ea bohloko: Ho fokotsa bohloko bo sa feleng.
(3) anti-rumbatory: Phokotso ea ho ruruha.
(4) Ho feto-fetoha ha ho fetoloa ha sesole sa 'mele.
(5) Neuroprotection: E sebelisoa ka mekhoa ea hora ea neuroprotective.
Ts'ebetso ea tlhahiso ea siomonine hydrokedide e ka akaretsoa ka tsela e latelang:
Herb tokisetso ea Herb:Ho hloekisa le ho omisa thepa ea semela se tala.
Ho tlotsoa:U sebelisa lithunya joaloka ethanol ho ntša sebe sa semela.
TLHOKOMELISO:Ho lelekisa solvent ho tsepamisa mohopolo dikahare tsa sinnomenine.
Alkalization:Ho fetola PH ho fetolela Sinotane ho mofuta oa eona oa letsoai.
Ho ntšoa metsi a metsi a metsi:Ho itlhoekisa ka solvents joalo ka anisole kapa 1-heptanool.
Ho hlatsoa:Ho hlatsoa ho akheha ho tlosa litšila le lipapatso tsa solvent.
Acidimer:Ho fokotsa PH ho ea ho Preomina hydrokendide.
Crystallization:Ho theha likristale tsa Siomenine hydrokeride.
Karohano:Centrifugigining kapa ho faela ho arola likristale tse fumanoeng tharollo.
Ho omella:Ho tlosa mongobo o sa feleng ho tsoa likristale.
Milling:Ho chesa likristale tse omileng hore e se ke ea fihla phofo e ntle.
Ho siela:Ho netefatsa hore na karolo e tšoanang ea likarolo tsa karolo e tšoanang.
Taolo ea Boleng:TLHOKOMELISO ea bohloeki ba bohloeki, ho tsepamisa maikutlo le litekanyetso tsa likokoana-hloko.
Ho paka:Sterlile le ho boloka liphutheloana tse sireletsehileng bakeng sa ho ajoa.
Boloka: Boloka sebaka se pholileng, se omileng le se hloekileng, se sireletse le mongobo le leseli le tobileng.
Package ea bongata: 25kg / moqomo.
Nako ea lead: matsatsi a 7 kamora odara ea hau.
Shel Life: Lilemo tse 2.
TLHOKOMELISO: Litlhaloso tse hlophiselitsoeng le tsona li ka fihleloa.
Express
Tlas'a 100kg, 3-5days
Ntlo ea PUSO EA PUSO SIRELETSO HO ETSA LINTHO TSE KHOLO
Ka leoatle
Ho feta300kg, matsatsi a ka bang 30
Port ho Port Port Travense Social Broker e hlokahalang
Ka moea
100Kg-1000kg, 5-7 Matsatsi a 5-7
Boema-fofane ho ea Boema-fofane ba Boema-fofane ba Coupleen e hlokahalang
BIOWA ORIC Orda o na le USDA le E NEST, BCC, ISO, Halal, Khese, ATLAL

